Chimie Bioinorganique; Chimie Bioorganométallique; Medicaments anti-cancer; Etudes mécanistiques; Etudes structurales
Biancalana Lorenzo, Gruchała Martyna, Batchelor Lucinda K., Błauż Andrzej, Monti Andrea, Pampaloni Guido, Rychlik Błażej, Dyson Paul J., Marchetti Fabio (2020), Conjugating Biotin to Ruthenium(II) Arene Units via Phosphine Ligand FunctionalizationConjugating Biotin to Ruthenium(II) Arene Units via Phosphine Ligand Functionalization, in
European Journal of Inorganic Chemistry, 2020(11-12), 1061-1072.
SchochSylvia, BatchelorLucinda K., FunaioliTiziana, CiancaleoniGianluca, ZacchiniStefano, BracciniSimona, ChielliniFederica, BiverTarita, PampaloniGuido, DysonPaul J., MarchettiFabio (2020), Diiron Complexes with a Bridging Functionalized Allylidene Ligand: Synthesis, Structural Aspects, and Cytotoxicity, in
Organomettalics, 39, 361-373.
Rocco Dalila, Batchelor Lucinda K., Ferretti Eleonora, Zacchini Stefano, Pampaloni Guido, Dyson Paul J., Marchetti Fabio (2020), Piano Stool Aminoalkylidene‐Ferracyclopentenone Complexes from Bimetallic Precursors: Synthesis and Cytotoxicity Data, in
ChemPlusChem, 85(1), 110-122.
Batchelor Lucinda K., De Falco Louis, Erlach Thibaud, Sharma Deepti, Adhireksan Zenita, Roethlisberger Ursula, Davey Curt A., Dyson Paul J. (2019), Crosslinking Allosteric Sites on the Nucleosome, in
Angewandte Chemie International Edition, 58(44), 15660-15664.
Rocco Dalila, Batchelor Lucinda K., Agonigi Gabriele, Braccini Simona, Chiellini Federica, Schoch Silvia, Biver Tarita, Funaioli Tiziana, Zacchini Stefano, Biancalana Lorenzo, Ruggeri Marina, Pampaloni Guido, Dyson Paul J., Marchetti Fabio (2019), Anticancer Potential of Diiron Vinyliminium Complexes, in
Chemistry – A European Journal, 25(65), 14801-14816.
Batchelor Lucinda K., Ortiz Daniel, Dyson Paul J. (2019), Histidine Targeting Heterobimetallic Ruthenium(II)–Gold(I) Complexes, in
Inorganic Chemistry, 58(4), 2501-2513.
Biancalana Lorenzo, Batchelor Lucinda K., Dyson Paul J., Zacchini Stefano, Schoch Silvia, Pampaloni Guido, Marchetti Fabio (2018), α-Diimine homologues of cisplatin: synthesis, speciation in DMSO/water and cytotoxicity, in
New Journal of Chemistry, 42(21), 17453-17463.
Biancalana Lorenzo, Batchelor Lucinda K., Funaioli Tiziana, Zacchini Stefano, Bortoluzzi Marco, Pampaloni Guido, Dyson Paul J., Marchetti Fabio (2018), α-Diimines as Versatile, Derivatizable Ligands in Ruthenium(II) p -Cymene Anticancer Complexes, in
Inorganic Chemistry, 57(11), 6669-6685.
Laurent Quentin, Batchelor Lucinda K., Dyson Paul J. (2018), Applying a Trojan Horse Strategy to Ruthenium Complexes in the Pursuit of Novel Antibacterial Agents, in
Organometallics, 37(6), 915-923.
Biancalana Lorenzo, Batchelor Lucinda K., Ciancaleoni Gianluca, Zacchini Stefano, Pampaloni Guido, Dyson Paul J., Marchetti Fabio (2018), Versatile coordination of acetazolamide to ruthenium( ii ) p -cymene complexes and preliminary cytotoxicity studies, in
Dalton Transactions, 47(28), 9367-9384.
Davey Gabriela E., Adhireksan Zenita, Ma Zhujun, Riedel Tina, Sharma Deepti, Padavattan Sivaraman, Rhodes Daniela, Ludwig Alexander, Sandin Sara, Murray Benjamin S., Dyson Paul J., Davey Curt A. (2017), Nucleosome acidic patch-targeting binuclear ruthenium compounds induce aberrant chromatin condensation, in
Nature Communications, 8(1), 1575-1575.
Batchelor Lucinda K., Păunescu Emilia, Soudani Mylène, Scopelliti Rosario, Dyson Paul J. (2017), Influence of the Linker Length on the Cytotoxicity of Homobinuclear Ruthenium(II) and Gold(I) Complexes, in
Inorganic Chemistry, 56(16), 9617-9633.
Adhireksan Zenita, Palermo Giulia, Riedel Tina, Ma Zhujun, Muhammad Reyhan, Rothlisberger Ursula, Dyson Paul J., Davey Curt A. (2017), Allosteric cross-talk in chromatin can mediate drug-drug synergy, in
Nature Communications, 8, 14860-14860.
Biancalana Lorenzo, Batchelor Lucinda K., De Palo Alice, Zacchini Stefano, Pampaloni Guido, Dyson Paul J., Marchetti Fabio (2017), A general strategy to add diversity to ruthenium arene complexes with bioactive organic compounds via a coordinated (4-hydroxyphenyl)diphenylphosphine ligand, in
Dalton Transactions, 46(36), 12001-12004.
En s’inspirant d’études précédentes, nous avons l’intention de développer des nouveaux agents thérapeutiques, conçus grâce aux informations obtenues de données cristallographiques et computationnelles. Une approche « atome-à-cellule » sera utilisée, comprenant des études structurales (cristallographie) et mécanistiques (computationnelles). Basé sur cette étude, nous devrions établir de nouveaux concepts pour améliorer et mieux contrôler la liaison de l’agent thérapeutique à sa cible.